opioid receptor — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T12314	Opioid receptor modulator 1		Opioid Receptor
	Opioid receptor modulator 1 is a modulator of opioid receptor.		Opioid Receptor
T9459	GR103545		Others
	GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.		Others
TP1832	Gluten Exorphin C		Opioid Receptor
	Gluten exorphin C is an opioid peptide derived from wheat gluten. Its IC50 values are 40 μM and 13.5 μM for μ opioid and δ opioid activities in the GPI and MVD assays, respectively.Gluten Exorphin C, isolated from the pe...		Opioid Receptor
T8991	BMS986187		Opioid Receptor
	BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.		Opioid Receptor
T13414	ZT 52656A hydrochloride		Opioid Receptor
	ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.		Opioid Receptor
T4386	PZM21		Opioid Receptor
	PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).		Opioid Receptor
T4351	DAMGO	Dagol,DAGO,RX-783006	Opioid Receptor
	DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents. Possible analgesic agent due to μ-opiod receptor interaction.		Opioid Receptor
T4407	SR17018		Opioid Receptor
	SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.		Opioid Receptor
T8992	BMS986188		Opioid Receptor
	BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.		Opioid Receptor
T0918	Trimebutine	Mebutin	Opioid Receptor
	Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid agonist effects. It is marketed for the treatment of irritabl...		Opioid Receptor
T62673	Mu opioid receptor antagonist 5
	Mu opioid receptor antagonist 5 (compound NAP) is a selective mu opioid receptor (MOR) antagonist that crosses the blood-brain barrier (EC50: 1.14 nM, Ki: 0.37 nM). Mu opioid receptor antagonist 5 can be used to study op...
T62766	Mu opioid receptor antagonist 2
	Mu opioid receptor antagonist 2 (compound 25) is a potent and selective mu opioid receptor (MOR) antagonist that permeates the blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM). Mu opioid receptor antagonist 2 can be used...
T62768	Mu opioid receptor antagonist 4
	Mu opioid receptor antagonist 4 (compound 31) is a potent and selective mu opioid receptor (MOR) antagonist that permeates the blood-brain barrier (Ki: 0.38 nM, EC50: 0.38 nM). Mu opioid receptor antagonist 2 can be used...
T7748	Dermorphin TFA		Others , Opioid Receptor
	Dermorphin TFA is a new class of opioids-like peptides		Others , Opioid Receptor
T7218	Endomorphin 2		Opioid Receptor
	Endomorphins-2 (EM-2) could decrease both the frequency and amplitude of the sEPSC of the motoneurons in lamina IX, which was reversed by the MOR antagonist CTOP. EM-2-IR fibers originated from primary afferent fibers f...		Opioid Receptor
T61901	σ1 Receptor/μ Opioid receptor modulator 1
	σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM). Opioid receptor modulator 1 shows potent analgesic activity, and ...
T4691	Asimadoline hydrochloride	EMD-61753 hydrochloride	Opioid Receptor
	Asimadoline hydrochloride (EMD-61753 hydrochloride) is a κ-opioid receptor agonist potentially for the treatment of pruritus. Asimadoline hydrochloride has also been shown to be used in the treatment of irritable bowel s...		Opioid Receptor
T79430	μ opioid receptor agonist 3		Opioid Receptor
	Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM. It holds promise for research into pain management and neuropsychiatric disorders [1].		Opioid Receptor
T62767	Mu opioid receptor antagonist 3
	Mu opioid receptor antagonist 3 (compound 26) is a potent and selective mu opioid receptor (MOR) antagonist that penetrates the blood-brain barrier (Ki: 0.24 nM, EC50: 0.54 nM). Mu opioid receptor antagonist 2 can be use...
T62025	μ opioid receptor agonist 2
	μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.